A. K. Ganguly Patents and Publications

A. K. Ganguly Patents and Publications

Books Published

Pramanik, Birendra N.; Ganguly, A.K.; Gross, Michael, L.   Applied Electrospray Mass Spectrometry . Marcel Dekker. New York 2002.

Shah, U.; Chackalamannil, S.; Ganguly, A.K.   Total Synthesis of Galbulimima  Alkaloids:  Himgaline and GB13  . Verlag-DM. 2008.

Patents

  1. Peptides as NS3-serine protease inhibitors of Hepatitis C Virus, U.S. Patent E043298 (2012)

  2. Human Immunodeficiency Virus Protease Inhibitors, U.S. Patent 20110112068 (2011)

  3. Preparation of Peptides as NS3-serine protease inhibitors of Hepatitis C Virus, U.S. Patent 2007032433 (2007)

  4. Preparation of Peptides as NS3-serine protease inhibitors of Hepatitis C Virus, U.S. Patent 2003216325 (2003)
  5. Ribavirin-Interferon Alpha Combination Therapy For Eradicating Detectable Hcv-Rna In Patients Having Chronic Hepatitis C Infection. U.S. Patent 2003004119 (2003).
  6. Monomeric Lipophilic Oligosaccharide Antibiotic Compositions. U.S. Patent 6380172 (2002).

  7. Preparation Of N-Imidazolylalkyl Piperazinecarboxamides As Inhibitors Of Farnesyl Protein Transferase. U.S. Patent 6,432,959 (2002).

  8. Ribavirin Derivative-Interferon-A Combination Therapy For Eradicating Detectable Hcv-Rna In Patients Having Chronic Hepatitis C Infection, And Preparation Of Ribavirin Derivatives. U.S. Patent 6,403,564 (2002).

  9. Preparation Of Amino Acid Esters Of Ribavirin For Hepatitis C Treatment. U.S. Patent 6277830 (2001).

  10. Tetrahydrofuran Antifungal Phosphate, Preparation Thereof, And Pharmaceutical Compositions. U.S. Patent 6,043,245(2000).

  11. Method For Treating Proliferative Diseases Using A Farnesyl Protein Transferase Inhibitor In Conjunction With An Antineoplastic Agent And/Or Radiation Therapy. U.S. Patent 6,096,757 (2000).

  12. Quasielastic Light Scattering Method Of Determining Monomeric Drug Content. U.S. Patent 5,948,688 (1999).

  13. Crystalline Interferon Alpha For Pulmonary Delivery And Method For Producing The Same, U.S. Patent 5,972,331 (1999).

  14. Method Of Determining Monomeric Drug Content, U.S. Patent 5,948,688 (1999).

  15. Water Soluble Antibiotics, U.S. Patent 5,795,874 (1998).

  16. Substituted Oximes, Hydrazones And Olefins As Neurokinin Antagonists, U.S. Patent 5,840,725 (1998).

  17. Oligosaccharide Antibiotics And Process For Preparation Thereof, U.S. Patent 5,763,600 (1998).

  18. Substituted Oximes, Hydrazones And Olefins As Neurokinin Antagonists, U.S. Patent 5,696,267 (1997).

  19. Tetrahydrofuran Antifungals, U.S. Patent 5,661,151 (1997).

  20. Benzo[5,6]Cycloheptapyridines, Compositions And Methods Of Use, U.S. Patent 5,665,726 (1997).

  21. Water Soluble Antibiotics, U.S. Patent 5,652,226 (1997).

  22. Nikkomycin Analogs, U.S. Patent 5,618,793 (1997).

  23. Orally Active Antiviral Compounds, U.S. Patent 5,618,849 (1997).

  24. Anti-Hiv (Aids) Agents, U.S. Patent 5,516,784 (1996).

  25. Pharmaceutically Active Compounds, U.S. Patent 5,459,144 (1995).

  26. Nikkomycin Analogs, U.S. Patent 5,461,055 (1995).

  27. Pharmaceutically Active Compounds, U.S. Patent 5,459,144 (1995).

  28. Imidazolyl Or Imidazoylalkyl Substituted With A Four Or Five Membered Nitrogen Containing Heterocyclic Ring, U.S. Patent 5,463,074 (1995).

  29. 2,2 Disubstituted Glycerol And Glycerol-Like Compounds, Compositions And Methods Of Use, U.S. Patent 5,449,680 (1995).

  30. Benzoalkano Compounds And Their Use For Treating Hyper-Proliferative Diseases, U.S. Patent 5,446,069 (1995).

  31. Benzo(5,6)Cycloheptapyridines, Compositions And Methods Of Use, U.S. Patent 5,438,062 (1995).

  32. Certain Substituted Phenoxy-Methyl Phenyl-Methoxy Benzenes Having Antiviral Activity, U.S. Patent 5,350,772 (1994).

  33. Anti-Fungal Uracil Compounds, U.S. Patent 5,346,898 (1994).

  34. 2,2-Disubstituted Glycerol And Glycerol-Like Compounds, Compositions And Methods Of Use, U.S. Patent 5,185,334 (1993).

  35. Pharmaceutically Active Compounds, U.S. Patent 5,272,167 (1993).

  36. Anti-Fungal Agents, U.S. Patent 5,238,926 (1993).

  37. Anti-Fungal Agents, U.S. Patent 5,236,900 (1993).

  38. Aryl Substituted Naphthalene Derivatives, U.S. Patent 5,225,436(1993).

  39. Processes For Preparing Bicyclic Compounds, U.S. Patent 5,180,823 (1993).

  40. Polycyclic Quinoline, Naphthyridine And Pyrazinopyridine Derivatives, U.S. Patent 5,126,352 (1992).

  41. Polycyclic Quinoline, Naphthyridine And Pyrazinopyridine Derivatives, U.S. Patent 5,116,840 (1992).

  42. Benzopyrido Piperidine, Piperidylidene And Piperazine Compounds, Compositions, Methods Of Manufacture And Methods Of Use, U.S. Patent 5,104,876 (1992).

  43. Benzo (5,6)Cycloheptapyridine Compounds, Compositions And Method Of Treating Allergies, U.S. Patent 5,089,496 (1992).

  44. Processes For Preparing Bicyclic Compounds And Intermediates Thereof, U.S. Patent 5,079,360 (1992).

  45. Fused Polycyclic Pyranyl Compounds As Antiviral Agents, U.S. Patent 5,034,531 (1991).

  46. Cyclic Diesters Of 4-Hydroxy-1,3-Benzenedimethanol And Compositions And Methods Employing Such Compounds, U.S. Patent 5,011,845 (1991).

  47. Process For Preparing Cyclopentyl Purine Derivatives, U.S. Patent 4,999,428 (1991).

  48. Polycyclic Quinoline, Naphthyridine And Pyrazinopyridine Derivatives, U.S. Patent 4,988,705 (1991).

  49. Process For Preparing Intermediates For Pharmaceutically Useful Bicyclic Compounds, U.S. Patent 4,897,487 (1990).

  50. Antiallergic 6,11-Dihydro-11-(4-Piperidylidene)-5h-Benzo

  51. (5,6)Cyclohepta(1,2-B)Pyridines, U.S. Patent 4,804,666 (1989).

  52. Pharmaceutically Active Compounds, U.S. Patent 4,851,423 (1989).

  53. 6,11-Dihydro-11-(N-Substituted-4-Piperidylidene)-5h-Benzo

  54. (5,6)Cyclohepta(1,2-B)Pyridines And Compositions And Methods Of Use, U.S. Patent 4,826,853 (1989).

  55. 6-Hydroxyethyl-2-Substituted Thio-Penem-3-Carboxylates, U.S. Patent 4,814,442 (1989).

  56. Polycyclic Quinoline, Naphthyridine And Pyrazinopyridine Derivatives, U.S. Patent 4,810,708 (1989).

  57. 2,4,4-Tri- And 2,2,4,4-Tetra Substituted-1,3-Dioxolane Antifungal, Antiallergy Compounds. U.S. Patent 4,788,190 (1988).

  58. Antibacterial 2-(Azacycloalkyl)Penems, U.S. Patent 4,743,598 (1988).

  59. 2-(Heterocycloalkylthio)Penems, U.S. Patent 4,690,922 (1987).

  60. Substituted Oligosaccharide Antibiotics, U.S. Patent 4,622,314 (1986).

  61. 2(N-Heterocyclyl)Penems, U.S. Patent 4,617,300 (1986).

  62. 2-(N-Heterocycloaliphaticthio)Penems, U.S. Patent 4,614,738 (1986).

  63. Heterocyclic Substituted Penems, U.S. Patent 4,587,241 (1986).

  64. Process For The Production Of Penems, U.S. Patent 4,584,133 (1986).

  65. Hydrazone Substituted Penems, U.S. Patent 4,559, 333 (1985).

  66. Processes For The Production Of Penems, U.S. Patent 4,530,793 (1985).

  67. 5r,6s,8r-6-(1-Hydroxyethyl)-2-(2-Carbamoyloxyethylthio)-Penem-3-Carboxylic Acid, U.S. Patent 4,504,485 (1985).

  68. Oxime Substituted Penems, U.S. Patent 4,503,064 (1985).

  69. Process For The Production Of Antibiotic Penems, U.S. Patent 4,443,373 (1984).

  70. 23-Demycinosyltylosin Compounds, Pharmaceutical Compositions And Method Of Use, U.S. Patent 4,436,729 (1984).

  71. 5r,6s,8r-2-(1-Methyl-2-Imidazolylmethylthio)-6-(1-Hydroxy-Ethyl)-Penem-3-Carboxylic Acid, U.S. Patent 4,435,412 (1984).

  72. Tylosin 20-Imino-20-Deoxo-4"-Acyl Derivatives, Pharmaceutical Compositions And Method Of Use, U.S. Patent 4,435,388 (1984).

  73. 6-(Hydroxyethyl)-2-[(Heterocyclyl Or Aryl)Thioalkylthio]-Penem-3-Carboxylates, U.S. Patent 4,431,654 (1984).

  74. Macrolide Antibacterial Ar-5 Components, U.S. Patent 4,373,095 (1983).

  75. (5r,6s,8r)-6-(1-Hydroxyethyl)-2-(2-Fluoroethylthio)-Penem-3-Carboxylates, U.S. Patent 4,411,906 (1983).

  76. Derivatives Of Antibiotic Ar-5 Components, U.S. Patent 4,366,309 (1982).

  77. 6-(Nitrogen-Containing Heterocyclic) Hydroxymethyl Penicillanic Acids, Compounds Related Thereto And Processes For Their Preparation, U.S. Patent 4,304,779 (1981).

  78. Synthesis Of ß-Lactams Having A Substituted Hydroxymethylene Group At The Position  Α To The Lactam Carbonyl Group, U.S. Patent 4,283,531 (1981).

  79. 6-(Substituted-Hydroxymethylene Penams), U.S. Patent 4,272,439 (1981).

  80. Novel 20-Imino Macrolide Antibacterial Agents, U.S. Patent 4,279,896 (1981).

  81. Amino Everninomicin And Derivatives Thereof, U.S. Patent 4,129,720.

  82. Triazolo [4,5-D]-Pyrimidines, U.S. Patent 4,076,711.

  83. Method Of Using Reduction Products Of Everninomicins As Antibacterial Agents And Pharmaceutical Compositions Useful Therefore, U.S. Patent 4,006,225.

  84. Electrochemical Process For Preparing Hydroxylaminoever-Ninomicins, U.S. Patent 3,998,708.

  85. Preparation Of 12, 13-Desepoxy-12,13-Dehydrorosamicin, U.S. Patent 3,975,372.

  86. Desevernitrose Everninomicins And Method For Their Manufacture, U.S. Patent 3,920,629.

  87. Reduction Products Of Everninomicins And Methods For Their Manufacture, U.S. Patent 3,915,956.

  88. Method Of Treating Fungal Infections With Azido Compounds, U.S. Patent 3,896,220.

  89. Process For The Preparation Of Rifamycin S And Analogs Thereof From The Halomicins, U.S. Patent 3,880,839.

  90. Azido Analogs Of Griseofulvin, U.S. Patent 3,816,472.

Publications

  1. Design, Synthesis, and X-ray Crystallographic Analysis of a Novel Class of HIV-1 Protease Inhibitors, Journal of Medicinal Chemistry 2011, 54, 7176-7183

  2. A convenient enantioselective synthesis of 3-asymmetrically substituted oxindoles as progesterone receptor antagonists, Tetrahedron Letters 52 (2011) 3945–3948

  3. 2-Phenylimidazo[1,2- b ]pyridazine derivatives highly active against  Haemonchus contorts , Bioorganic & Medicinal Chemistry Letters 21 (2011) 4160–4163

  4. Synthesis and Atropisomerism of 2,2'- ortho  Disubstituted Biphenyls, Tetrahedron Letters, 51 6213-6215. 2010

  5. Synthesis of Conformationally Restricted Sulfonamides via  Radical Cyclisation, Tetrahedron Letters, 51 2681-2684. 2010

  6. A Convenient Synthesis of  ortho-ortho  Disubstituted Biphenyls Containing an Eight-membered Lactam Ring Using Radical Chemistry, Tetrahedron Letters, 50 (17), 1879-1881. 2009
  7. (Posaconazole (Noxafil, SCH56592), a New Azole Antifungal Drug, Was a Discovery Based on the Isolation and Mass Spectral Characterization of a Circulating Metabolite of an Earlier Lead (SCH 51048), Journal of Mass Spectrometry, 43 509-517. 2008
  8. Mass Spectrometric Studies of Potent Inhibitors of Farnesyl Protein Transferase - Detection of Pentameric Noncovalent Complexes, Journal of Mass Spectrometry, 43 1393-1401. 2008
  9. Some Aspects of Medicinal Chemistry at the Schering-Plough Research Institute; Comprehensive Medicinal Chemistry II, 8:29 2007
  10. Total Synthesis of ( - )-Himgaline;  Journal of The American Chemical Society, 128 12654 July 20 2006

  11. Synthesis of Oxygen Heterocycles;  Tetrahedron Letters 47 (8): 1347-1349 Feb 20 2006

  12. Guiding Farnesyltransferase Inhibitors From An Eclips (R) Library To The Catalytic Zinc;  Bioorganic & Medicinal Chemistry Letters 16 (3): 507-511 Feb 1 2006

  13. Hydroxylated Analogues Of The Orally Active Broad Spectrum Antifungal, Sch51048 (1), And The Discovery Of Posaconazole [Sch 56592; 2 Or (S,S)-5] ; Bioorganic & Medicinal Chemistry Letters 16 (1): 186-190 Jan 1 2006

  14. Surfing The Piperazine Core Of Tricyclic Farnesyltransferase Inhibitors ; Bioorganic & Medicinal Chemistry Letters 15 (24): 5537-5543 Dec 15 2005

  15. Synthesis And Properties Of 3-Acyl-Gamma-Pyrones, A Novel Class Of Flavones  and Chromones;  Tetrahedron Letters 46 (23): 4119-4121 Jun 6 2005

  16. Structure Determination And Conformation Analysis Of Symmetrical Dimers ; Magnetic Resonance In Chemistry 43 (3): 187-199 Mar 2005

  17. Synthesis Of Highly Condensed Heterocycles Using Radical Reactions ; Tetrahedron Letters 45 (48): 8909-8912 Nov 22 2004

  18. Synthesis Of Heterocyclic Compounds Using Radical Reactions And Evidence For The Formation Of Spiro Radical Intermediates (Vol 45, Pg 883, 2004) ; Tetrahedron Letters 45 (19): 3835-3835 May 3 2004

  19. Drug Discovery At Schering-Plough Research Institute - A Few Case Studies. ; Abstracts Of Papers Of The American Chemical Society 225: U203-U203 167-Medi Part 2 Mar 2003

  20. Synthesis Of Heterocyclic Compounds Using Radical Reactions And Evidence For The Formation Of Spiro Radical Intermediates ; Tetrahedron Letters 45 (4): 883-886 Jan 19 2004

  21. 1h-Pyrazolo-[3,4-C]Cyclophepta[1,2-C]Thiophenes: A Unique Structural Class Of Dopamine D4 Selective Ligands, Bioorganic & Medicinal Chemistry Letters (2003), 13(17), 2921-4.

  22. A Highly Stereoselective Approach To Novel 2,2,4-Trisubstituted Pyrrolidines By Halocylization: Key Intermediates Towards Syntheses Of Nitrogen Analogs Of Noxafil (R) ; Tetrahedron Letters 44 (43): 7997-8000 Oct 20 2003

  23. Negative Ion Multiple-Stage Mass Spectrometric Analysis Of Complex  Oligosaccharides (Everninomicins) In A Quadrupole Ion Trap: Implications For  Charge-Remote Fragmentation ; Arkivoc : 31-44 Part 3 2003

  24. Trihalobenzocycloheptapyridine Analogues of Sch 66336 As Potent Inhibitors of Farnesyl Protein Transferase ; Bioorganic & Medicinal Chemistry 11 (1): 139-143 Jan 2 2003

  25. Solution- And Solid-Phase Synthesis Of Enantiomerically Pure Spiro Oxindoles ; Tetrahedron Letters 43 (49): 8981-8983 Dec 2 2002

  26. Synthesis Of Heterocyclic Compounds Using Radical Reactions ; Tetrahedron Letters 43 (38): 6865-6868 Sep 16 2002

  27. Pharmacology Of ;  N-(3,5-Dichloro-1-Oxido-4-Pyridinyl)-8-Methoxy-2-(Trifluoro- Methyl)-5-Quinoline Carboxamide (Sch 351591), A Novel, Orally Active Phosphodiesterase 4 Inhibitor ; Journal Of Pharmacology And Experimental Therapeutics 302 (1):127-137 Jul 2002

  28. 8-Methoxyquinolines As Pde4 Inhibitors ; Bioorganic & Medicinal Chemistry Letters 12 (12): 1617-1619 Jun 17 2002

  29. Synthesis And Profile Of Sch351591, A Novel Pde4 Inhibitor ; Bioorganic & Medicinal Chemistry Letters 12 (12): 1621-1623 Jun 17 2002

  30. Structural Characterization Of The Oligosaccharide Antibiotic Everninomicins By Positive And Negative Ion Esi And Fab Mass Spectrometry, Advances In Mass Spectrometry (2001), 15, 907-908.

  31. Farnesyl Protein Transferase Inhibition: A Novel Approach To Anti-Tumor Therapy. The Discovery And Development Of Sch 66336 ; Current Medicinal Chemistry 8 (12): 1419-1436 Oct 2001

  32. Discovery Of Potent, Orally Bioavailable Ccr5 Antagonists - 1. ; Abstracts Of Papers Of The American Chemical Society 221: 26-Medi Part 2 Apr 1 2001

  33. Discovery Of Potent, Orally Bioavailable Ccr5 Antagonists - 2. ; Abstracts Of Papers Of The American Chemical Society 221: 27-Medi Part 2 Apr 1 2001

  34. Enantioselective Syntheses Of Carbocyclic Ribavirin And Its Analogs: Linear  Versus Convergent Approaches Tetrahedron Letters 41 (49): 9575-9579 Dec 2 2000

  35. High-Resolution Lc/Ms For Analysis Of Minor Components In Complex Mixtures: Negative Ion Esi For Identification Of Impurities And Degradation Products Of a  Novel Oligosaccharide Antibiotic ; Journal Of Mass Spectrometry 35 (11): 1252-1258 Nov 2000

  36. Ziracin, A Novel Oligosaccharide Antibiotic ; Journal Of Antibiotics 53 (10): 1038-1044 Oct 2000

  37. Advancing The Frontiers Of Anticancer Therapy: Discovery Of The Farnesyl Protein Transferase Inhibitor Sch-66336. Abstracts Of Papers Of The American Chemical Society 219: 293-Medi Part 2 Mar 26 2000

  38. Synthesis And Biological Activity Of New  Piperazine-2-Carboxyamide-Halobenzocycloheptapyridine Heterocycles As  Inhibitors Of Ras Farnesyl Protein Transferase. ; Abstracts Of Papers Of The American Chemical Society 219: 305-Medi Part 2 Mar 26 2000

  39. Structural Characterization Of The Oligosaccharide Antibiotics Everninomicins By  Negative Ion Fab And Esi/Ms ; Journal Of Antibiotics 53 (6): 640-643 Jun 2000

  40. Synthesis Of C-11 Methyl-Substituted Benzocycloheptapyridine Inhibitors of  Farnesyl Protein Transferase ; Organic Letters 1 (9): 1371-1373 Nov 4 1999

  41. Discovery Of Indolocycloheptapyridine Inhibitors Of Farnesyl Protein Transferase By De Novo Analysis Of The X-Ray Crystal Structure Of Sch-66336-R-Fpt.; Abstracts Of Papers Of The American Chemical Society 218:; 165-Medi Part 1 Aug 22 1999

  42. Tricyclic Farnesyl Protein Transferase Inhibitors: Crystallographic And Calorimetric Studies Of Structure-Activity Relationships. ; Abstracts Of Papers Of The American Chemical Society 218: 209-Medi Part 1 Aug 22 1999

  43. Identification Of Pharmacokinetically Stable 3,10-Dibromo-8-Chlorobenzocycloheptapyridine Farnesyl Protein Transferase Inhibitors With Potent Enzyme And Cellular Activities Journal Of Medicinal Chemistry 42 (14): 2651-2661 Jul 15 1999

  44. Tricyclic Farnesyl Protein Transferase Inhibitors: Crystallographic And Calorimetric Studies Of Structure-Activity Relationships ; Journal Of Medicinal Chemistry 42 (12): 2125-2135 Jun 17 1999

  45. Atropisomeric Trihalobenzocycloheptapyridine Analogues Provide Stereoselective Fpt Inhibitors With Antitumor Activity ; Bioorganic & Medicinal Chemistry 7 (5): 861-867 May 1999

  46. Chemical Modifications And Structure Activity Studies Of Ziracin And Related Everninomicin Antibiotics ; Bioorganic & Medicinal Chemistry Letters 9 (8): 1209-1214 Apr 19 1999

  47. An Introduction To Electrospray Ionization And Matrix Assisted Laser Desorption/Ionization Mass Spectrometry: Essential Tools In The Modern Drug Discovery Process ; Journal Of The Indian Chemical Society 75 (10-12): 621-627 Oct-Dec 1998

  48. Dual Antagonists Of Platelet Activating Factor And Histamine - 3. Synthesis, Biological Activity And Conformational Implications Of Substituted N-Acyl-Bis-Arylcycloheptapiperazines.;  Bioorganic & Medicinal Chemistry Letters 8 (24): 3469-3474 Dec 15 1998

  49. Interaction Of A Novel Gdp Exchange Inhibitor With The Ras Protein; Biochemistry 37 (45): 15631-15637 Nov 10 1998

  50. (+)-4-[2-[4-(8-Chloro-3,10-Dibromo-6,11-Dihydro-5h-Benzo[5,6]Cyclohepta[1,2-B]-Pyridin-11(R)-Yl)-1-Piperidinyl]-2-Oxo-Ethyl]-1-Piperidinecarboxamide (Sch-66336): A Very Potent Farnesyl Protein Transferase Inhibitor As A Novel Antitumor Agent ; Journal Of Medicinal Chemistry 41 (24): 4890-4902 Nov 19 1998

  51. Electrospray Ionization Mass Spectrometry For The Study Of Non-Covalent Complexes: An Emerging Technology ; Journal Of Mass Spectrometry 33 (10): 911-920 Oct 1998

  52. Elucidation Of Sch 49088, A Novel Everninomicin Antibiotic Containing An Unusual Hydroxylamino-Ether Sugar, Everhydroxylaminose ; Tetrahedron Letters 39 (46): 8441-8444 Nov 12 1998

  53. Synthesis And Antibacterial Activity Of 2-Alkoxy Penems ; Bioorganic & Medicinal Chemistry Letters 8 (19): 2793-2796 Oct 6 1998

  54. Synthesis And Biological Activity Of Novel N-Cyanoguanidine-Halobenzocycloheptapyridine Heterocycles As Inhibitors Of Ras Farnesyl Protein Transferase. ; Abstracts Of Papers Of The American Chemical Society 216: 304-Medi Part 2 Aug 23 1998

  55. Potent, Selective, And Orally Bioavailable Tricyclic Pyridyl Acetamide N-Oxide Inhibitors Of Farnesyl Protein Transferase With Enhanced In Vivo Antitumo; R journal Of Medicinal Chemistry 41 (10): 1561-1567 May 7 1998

  56. Structural Elucidation Of Ziracin, A Novel Antibiotic Which Is Active Against Organisms Resistant To Methicillin And Vancomycin ; Journal Of The Indian Chemical Society 74 (11-12): 980-986 Nov-Dec 1997

  57. One Pot Solid Phase Synthesis Of Isoxazolines ; Tetrahedron Letters 39 (17): 2447-2448 Apr 23 1998

  58. Inhibitors Of Farnesyl Protein Transferase. 4-Amido, 4-Carbamoyl, And 4-Carboxamido Derivatives Of 1-(8-Chloro-6,11-Dihydro-5h-Benzo[5,6]Cyclohepta- [1,2-B]Pyridin-11-Yl)Piperazineand1-(3-Bromo-8-Chloro-6,11-Dihydro-5h-Benzo [5,6]Cyclohepta[1,2-B]Pyridin-11-Yl)Piperazine ; Journal Of Medicinal Chemistry 41 (6): 877-893 Mar 12 1998

  59. Orally Active, Trihalobenzocycloheptapyridine Farnesyl Protein Transferase Inhibitor Antitumor Agents. ; Abstracts Of Papers Of The American Chemical Society 215: 102-Medi Part 1 Apr 2 1998

  60. Highly Regioselective Nitration Reactions Provide A Versatile Method Of Functionalizing Benzocycloheptapyridine Tricyclic Ring Systems: Application Toward Preparation Of Nanomolar Inhibitors Of Farnesyl Protein Transferase ; Journal Of Organic Chemistry 63 (3): 445-451 Feb 6 1998

  61. Trans-4-Methyl-3-Imidazoyl Pyrrolidine As A Potent, Highly Selective Histamine H-3 Receptor Agonist In Vivo ; Bioorganic & Medicinal Chemistry Letters 8 (3): 243-248 Feb 3 1998

  62. Structure-Activity Relationship Of 3-Substituted N-(Pyridinylacetyl)-4-(8-Chloro-5,6-Dihydro-11h-Benzo[5,6]Cyclohepta[1,2-B]Pyridin-11-Ylidene)-Piperidine Inhibitors Of Farnesyl-Protein Transferase: Design And Synthesis Of In Vivo Active Antitumor Compounds ; Journal Of Medicinal Chemistry 40 (26): 4290-4301 Dec 19 1997

  63. Determination Of The Absolute Stereochemistry At The C16 Orthoester Of Everninomicin Antibiotics; A Novel Acid-Catalyzed Isomerization Of Orthoesters ; Tetrahedron Letters 38 (46): 7989-7992 Nov 17 1997

  64. Structure Elucidation Of Everninomicin-6, A New Oligosaccharide Antibiotic, By Chemical Degradation And Fab-Ms Methods ; Journal Of The American Society For Mass Spectrometry 8 (11): 1134-1140 Nov 1997

  65. Elucidation Of A Ras-Inhibitor Complex By Ms, Nmr And Molecular Modeling ; Abstracts Of Papers Of The American Chemical Society 214: 204-Comp Part 1 Sep 7 1997

  66. Total Synthesis Of The Antifungal Cyclic Depsipeptides Sch 53174 And 54256 ; Abstracts Of Papers Of The American Chemical Society 214: 159-Medi Part 1 Sep 7 1997

  67. Inhibitors Of Farnesyl Protein Transferase .2. 4-Amino, 4-Carbamoyl And 4-Carboxamido Derivatives Of 1-(3-Bromo-8-Chloro-6,11-Dihydro-5h-Benzo[5,6]Cyclohepta[1,2-B]Pyridin-11-Yl)Piperazine. ; Abstracts Of Papers Of The American Chemical Society 214: 194-Medi Part 1 Sep 7 1997

  68. Complete H-1 And C-13 Nmr Assignments Of The Oligosaccharide Antibiotic Sch 27899 ; Magnetic Resonance In Chemistry 35 (8): 529-532 Aug 1997

  69. Detection And Structural Characterization Of Ras Oncoprotein-Inhibitors Complexes By Electrospray Mass Spectrometry ; Bioorganic & Medicinal Chemistry 5 (5): 817-820 May 1997

  70. Inhibitors Of Farnesyl Protein Transferase .1. 4-Amido, 4-Carbamoyl And 4-Carboxamido Derivatives Of 1-(8-Chloro-6,11-Dihydro-5h-Benzo(5,6) Cyclohepta(1,2-B) Pyridin-11-Yl)Piperazine. ; Abstracts Of Papers Of The American Chemical Society 213: 199-Medi Part 2 Apr 13 1997

  71. Recent Studies On Azoles; Discovery And Synthesis Of Sch 56592, A Broad Spectrum Orally Active Antifungal Agent. ; Abstracts Of Papers Of The American Chemical Society 213: 318-Medi Part 2 Apr 13 1997

  72. Antitumor 8-Chlorobenzocycloheptapyridines: A New Class Of Selective, Nonpeptidic, Nonsulfhydryl Inhibitors Of Ras Farnesylation ; Bioorganic & Medicinal Chemistry 5 (1): 93-99 Jan 1997

  73. Discovery Of Novel Nonpeptide Tricyclic Inhibitors Of Ras Farnesyl Protein Transferase ; Bioorganic & Medicinal Chemistry 5 (1): 101-113 Jan 1997

  74. Ras Oncoprotein Inhibitors: The Discovery Of Potent, Ras Nucleotide Exchange Inhibitors And The Structural Determination Of A Drug-Protein Complex ; Bioorganic & Medicinal Chemistry 5 (1): 125-133 Jan 1997

  75. Novel Tricyclic Aminoacetyl And Sulfonamide Inhibitors Of Ras Farnesyl Protein Transferase ; Bioorganic & Medicinal Chemistry Letters 6 (24): 2977-2982 Dec 17 1996

  76. Concise Asymmetric Routes To 2,2,4-Trisubstituted Tetrahydrofurans Via Chiral Titanium Imide Enolates: Key Intermediates Towards Synthesis Of Highly Active Azole Antifungals Sch 51048 And Sch 56592 (Vol 37, Pg 5657, 1996) ; Tetrahedron Letters 37 (38): 6821-6821 Sep 16 1996

  77. Concise Asymmetric Routes To 2,2,4-Trisubstituted Tetrahydrofurans Via Chiral Titanium Imide Enolates: Key Intermediates Towards Synthesis Of Highly Active Azole Antifungals Sch 51048 And Sch 56592 l; Tetrahedron Letters 37 (32): 5657-5660 Aug 5 1996

  78. Total Synthesis Of The Antifungal Cyclic Depsipeptides Sch 57697 And Aureobasidin A ; Tetrahedron Letters 37 (32): 5661-5664 Aug 5 1996

  79. Synthesis Of An Optically Pure 3-Unsubstituted Beta-Lactam Using An Asymmetric Reformatsky Reaction And Its Conversion To Cholesterol Absorption Inhibitors ; Tetrahedron Letters 37 (24): 4095-4098 Jun 10 1996

  80. Ras Oncoprotein Inhibitors: The Discovery Of Potent, Ras Nucleotide Exchange Inhibitors And The Structure Determination Of A Drug-Protein Complex. Abstracts Of Papers Of The American Chemical Society 211: 87-Medi Part 2 Mar 24 1996

  81. Sch 51048, A Novel Broad-Spectrum Orally Active Antifungal Agent: Synthesis And Preliminary Structure-Activity Profile, Bioorganic & Medicinal Chemistry Letters, Vol. 5, No. 2, 127-132, 1995.

  82. An Enantioselective Synthesis Of The Antifungal Agent (2r,3r)-2-(2,4-Difluorophenyl)-3-(Methylsulfonyl)-1-(1,2,4-Triazol-1-Yl)-2-Butanol (Sch-42427, Sm-9164) ; Synlett (11): 1110& Nov 1995

  83. A Novel Pyrrolidine Analog Of Histamine As A Potent, Highly Selective Histamine H-3 Receptor Agonist ; Journal Of Medicinal Chemistry 38 (10): 1593-1599 May 12 1995

  84. Highly Stereoselective Access To Novel 2,2,4-Trisubstituted Tetrahydrofurans By Halocyclization - Practical Chemoenzymatic Synthesis Of Sch-51048, A Broad-Spectrum Orally-Active Antifungal Agent ; Tetrahedron Letters 36 (11): 1787-1790 Mar 13 1995

  85. Enantioselective Synthesis Of The Optical Isomers Of Broad-Spectrum Orally Active Antifungal Azoles, Sch 42538 And Sch 45012, Bioorganic & Medicinal Chemistry Letters, Vol. 4, No. 16, 2023-2028, 1994.

  86. The Synthesis Of Novel Hiv-Protease Inhibitors, Bioorganic & Medicinal Chemistry, Vol. 2, No. 10, Pp. 1075-1083, 1994.

  87. Indolocarbazole Nitrogens Linked By Three-Atom Bridges: A Potent New Class Of Pkc Inhibitors, Bioorganic & Medicinal Chemistry Letters, Vol. 4, No. 11, Pp 1333-1338, 1994.

  88. Synthesis Of Novel Azole Antifungals By A Modified Sharpless Asymmetric Dihydroxylation, Synlett, No. 4, P 263, 1994.

  89. The Synthesis Of Novel Hiv-Protease Inhibitors Via Silica Gel Assisted Addition Of Amines To Epoxides, Synlett, No. 9, P. 703, 1993.

  90. A Cyclization-Trapping Route To Carbocyclic And Heterocyclic Benzylic Sulfones, Tetrahedron Letters, Vol. 34, No. 50, 8033-8036, 1993.

  91. Penems Containing Amino Acid Derived Substituents At C-2, Bioorganic & Medicinal Chemistry Letters, Vol. 3, No. 11, 2177-2182, 1993.

  92. Controlling Benzylic And Anomeric Functionality And Stereochemistry: Methodology And Syntheses Utilising Intramolecular Ionic Hydrogenation, Synlett, Accounts & Rapid Communications In Synthetic Organic Chemistry, No. 8, Pp 541-547, August 1993.

  93. Application Of Electrospray Mass Spectrometry In Probing Protein-Protein And Protein-Ligand Noncovalent Interactions, J. Am. Soc. Mass Spectrom., 4, 624-630 1993.

  94. Indolocarbazoles-Ii. Synthetic Studies Towards Staurosporine. An Unexpected 1,2 Migration Of Indolocarbazole Nitrogen Results In A Novel And Potent Protein Kinase C Inhibitor, Tetrahedron Letters, Vol. 34, No. 36, Pp. 5685-5688, 1993.

  95. Studies Of The Ras-Gdp And Ras-Gtp Noncovalent Complexes By Electrospray Mass Spectrometry, Tetrahedron, Vol. 49, No. 36, Pp. 7985-7996, 1993.

  96. A Synthesis Of Nikkomycin Z: Improved Synthesis And Protection Of The Pyridyl  Γ -Hydroxy-Α-Aminobutanoic Acid Component, Tetrahedron Letters, Vol. 34, No. 20, Pp 326 7-3270, 1993.

  97. A Convenient Degradation Of Polyoxin D To Uracil Polyoxin C: Access To Key Intermediates And Synthesis Of Antifungal Α-Aminoacyl Derivatives Of Upoc, Bioorganic & Medicinal Chemistry Letters, Vol. 3, No. 6, Pp 1079-1084, 1993.

  98. Dual Antagonists Of Platelet Activating Factor And Histamine. 2. Pyridine Ring Substitution Of N-Acetyl-4-(8-Chloro-5,6-Dihydro-11h-Benzo[5,6]Cyclohepta[1,2-B]Pyridin-11-Ylidene)Piperidines, Bioorganic & Medicinal Chemistry Letters, Vol. 3, No. 6, Pp 1073-1078, 1993.

  99. Structure Determination Of Antiviral Compound Sch 38057 Complexed With Human Rhinovirus 14, J. Mol. Biol. 230, 857-867, 1993.

  100. Total Synthesis And Absolute Stereochemistry Of The Antifungal Dipeptide Sch 37137 And Its 2s,3s-Isomer, Tetrahedron Letters, Vol. 34, No. 20, Pp 3201-3204, 1993.

  101. A Synthesis Of Nikkomycin Z: Improved Synthesis And Protection Of The Pyridyl   -Hydroxy-Α-Aminobutanoi c Acid Component, Tetrahedron Letters, Vol. 34, No. 20, Pp 3267-3270, 1993.

  102. Aqueous Diels-Alder Reactions Of Electron Deficient 2-Arylfurans: A Highly Stereoselective Route To 2,2,5-Trisubstituted Tetrahydrofurans Towards A Novel Class Of Orally Active Azole Antifungals, Heterocycles, Vol. 35, No. 1, 1993.

  103. Ring Contraction Reactions Of 2-O-Methanesulfonates Of Alpha-Hydroxy-Gamma-Lactones In Aqueous-Medium To Oxetane-2-Carboxylic Acids – A Convenient Synthesis Of 3'-O-Methyloxetanocin And A Formal Synthesis Of Oxetanocin ; Tetrahedron Letters 33 (50): 7721-7724 Dec 8 1992

  104. Biology And Synthesis Of Sch-40120, An Antipsoriatic Agent That Inhibits 5-Lipoxygenation And T-Cell Proliferation ; Abstracts Of Papers Of The American Chemical Society 204: 2-Medi Part 1 Aug 23 1992

  105. Synthetic Studies On Nikkomycin X/Z - Synthesis Of The Pyridyl Amino-Acid Portion, And Peptide Coupling ; Abstracts Of Papers Of The American Chemical Society 204: 125-Orgn Part 2 Aug 23 1992

  106. A General Strategy For The Synthesis Of Antiviral Scopadulcic Acids ; Abstracts Of Papers Of The American Chemical Society 204: 307-Orgn Part 2 Aug 23 1992

  107. Mass-Spectrometric Detection Of The Noncovalent Gdp-Bound Conformational State Of The Human H-Ras Protein ; Journal Of The American Chemical Society 114 (16): 6559-6560 Jul 29 1992

  108. Synthesis Of (+)-8-Methyl Cercosporamide - Stereochemical Correlation Of Natural (-)-Cercosporamide With (+)-Usnic Acid ; Tetrahedron 48 (23): 4757-4766 Jun 5 1992

  109. Selective Transformations Of The Antifungal Antibiotic Polyoxin-D - Synthesis Of Peptide Derivatives With Chitin Synthetase-Activity ; Abstracts Of Papers Of The American Chemical Society 203: 62-Medi Part 2 Apr 5 1992

  110. Recent Studies On Veratrum Alkaloids: Selective Modifications Of Rings Def And Their Effect On Hypotensive/Emetic Activities, Xiith International Symposium On Medicinal Chemistry, Basel, Switzerland, September, 1992.

  111. Sch-40338, A New Dual Paf And Histamine Antagonist Related To Sch-37370 ; Abstracts Of Papers Of The American Chemical Society 202: 161-Medi Part 1 Aug 25 1991

  112. A Practical Conversion Of An Azetidinone To Penem - Synthesis Of Sch 34343 ; Tetrahedron 48 (7): 1175-1182 Feb 14 1992

  113. Antibiotics: Oligosaccharides, Kirk-Othmer Encyclopedia Of Chemical Technology - 4th Ed., Vol. No. 3, P. 259-266, 1992.

  114. Discovery And Preliminary Pharmacology Of Sch-37370, A Dual Antagonist Of Paf And Histamine ; Lipids 26 (12): 1172-1174 Dec 1991

  115. Synthesis Of The Antifungal Agent Sch-42427 (Sm-9164) ; Bioorganic & Medicinal Chemistry Letters 1 (7): 349-352 1991

  116. Isomer Differentiation And Structural Characterization Of Penem Beta-Lactam Antibiotics By Mass-Analyzed Ion Kinetic-Energy Spectrometry ; Organic Mass Spectrometry 26 (8): 703-708 Aug 1991

  117. Alkylation Of 2-Oxy-Substituted 1-Sulfonylallyl And 1-Sulfonylvinyl Anions – New Routes To Functionalized Carbocycles And Dihydrofurans ; Journal Of Organic Chemistry 56 (11): 3556-3564 May 24 1991

  118. Controlling Benzylic Functionality And Stereochemistry .1. Synthesis Of The Secopseudopterosin Aglycone  ; Tetrahedron Letters 32 (19): 2083-2086 May 6 1991

  119. Controlling Benzylic Functionality And Stereochemistry .2. Synthesis Of The Pseudopterosin Aglycone ; Tetrahedron Letters 32 (19): 2087-2090 May 6 1991

  120. Dual Antagonists Of Platelet-Activating-Factor And Histamine - Identification Of Structural Requirements For Dual Activity Of N-Acyl-4-(5,6-Dihydro-11h-Benzo[5,6]Cyclohepta-[1,2-B]Pyridin-11-Ylidene)Piperidines ; Journal Of Medicinal Chemistry 34 (1): 457-461 Jan 1991

  121. Macrolactams - A New Class Of Antifungal Agents ; Journal Of The American Chemical Society 112 (17): 6403-6405 Aug 15 1990

  122. Stereospecific Synthesis Of The Aglycone Of Pseudopterosin-E ; Pure And Applied Chemistry 62 (7): 1289-1291 Jul 1990

  123. Synthesis Of A New Series Of Dual Paf And Histamine-Antagonists ; Abstracts Of Papers Of The American Chemical Society 198: 56-Medi Sep 10 1989

  124. Structure-Activity Relationship Studies In A Series Of Dual Paf And Histamine-Antagonists ; Abstracts Of Papers Of The American Chemical Society 198: 88-Medi Sep 10 1989

  125. Hydroxylated Metabolites Of Loratadine - An Example Of Conformational Diastereomers Due To Atropisomerism ; Journal Of Organic Chemistry 55 (10): 3341-3350 May 11 1990

  126. Cyclofunctionalization Of Epoxyalcohol Derivatives .4. Cyclization Of Sulfonylacetate Dianions - A Synthesis Of Mebmt ; Tetrahedron Letters 30 (50): 7029-7032 1989

  127. A Concise Route To The Oxathiazepine Containing Eudistomin Skeleton And Some Carba-Analogs ; Tetrahedron Letters 30 (49): 6809-6812 1989

  128. Synthesis Of A Carbocyclic Analog Of Quercetin Via A Barbier Reaction ; Tetrahedron Letters 30 (41): 5563-5566 1989

  129. Synthesis Of 14-Alpha-Aminomethyl Substituted Lanosterol Derivatives – Inhibitors Of Fungal Ergosterol Biosynthesis ; Journal Of The Chemical Society-Chemical Communications (14): 898-900 Jul 15 1989

  130. Free-Radical Cyclization In The Synthesis Of Fused Bicyclic Beta-Lactams ; Heterocycles 28 (1): 47-49 Jan 1 1989

  131. The Structure Of New Oligosaccharide Antibiotics, 13-384 Component-1 And Component-5 ; Heterocycles 28 (1): 83-88 Jan 1 1989

  132. Ionization Of Penem Beta-Lactam Antibiotics Using Thermospray (Filament-On) Mass-Spectrometry ; Journal Of Antibiotics 41 (9): 1268-1271 Sep 1988

  133. Synthesis And Invitro Activity Of The Penem Antibiotics ; Medicinal Research Reviews 8 (3): 393-440 Jul-Sep 1988

  134. An Efficient Synthesis Of (3r,4r)-3-(1(R)-Hydroxyethyl)-4-(Benzoyloxy)-2-Azetidinone From L-Threonine - Use Of Phenylalkoxymethyl As A Novel N-Protecting Group ; Journal Of Organic Chemistry 53 (2): 450-452 Jan 22 1988

  135. A New Ring Synthesis For 3-Substituted And Polysubstituted Furans - Directing Effects Of A 3-(Arenesulfonyl) Group In Metalation And Friedel-Crafts Processes ; Tetrahedron Letters 28 (36): 4123-4126 1987

  136. Configurational Properties And Chemical-Reactivity Of Mono And Dianions Derived From Aryl 2-Alkoxyvinyl ; Sulfones ; Tetrahedron Letters 28 (36): 4127-4130 1987

  137. A Convenient Synthesis Of Polyoxamic Acid, 5-O-Carbamoylpolyoxamic Acid, And Their Unnatural D Isomers ; Journal Of Organic Chemistry 51 (25): 5024-5028 Dec 12 1986

  138. Fast-Atom-Bombardment Mass-Spectrometry - A Powerful Technique For Study Of Oligosaccharide Antibiotics ; Indian Journal Of Chemistry Section B-Organic Chemistry Including Medicinal Chemistry 25 (11): 1105-1111 Nov 1986

  139. A New Class Of 2-Heterocycyl-Alkylthiopenems; Journal Of Antibiotics 39 (8): 1182-1186 Aug 1986

  140. A New Class Of Penems-C-2-N-Substituted Compounds-Synthesis And Antibacterial Activity ; Journal Of Antibiotics 39 (8): 1187-1190 Aug 1986

  141. Cyclofunctionalization Of Epoxyalcohol Derivatives .1. Delivery Of Functionalized Carbon For Stereospecific Synthesis Of Dihydrofurans And Dihydroxyacids;  Tetrahedron Letters 26 (51): 6301-6304 1985

  142. Synthesis And Preliminary Invitro Profile Of Sch 34343 – A New Penem Antibacterial Agent ; Journal Of Antimicrobial Chemotherapy 15: 1-4 Suppl. C; 1985

  143. The Use Of Fast Atom Bombardment Mass-Spectrometry For The Determination Of Structures Of Everninomicins ; Journal Of Antibiotics 38 (6): 808-812 1985

  144. Synthesis Of Penem Antibiotics ; Heterocycles 21: 421-421 Sp. Iss. Si 1984

  145. Synthesis Of Penem Antibiotics, Recent Advances In The Chemistry Of ß-Lactam Antibiotics, Third International Symposium, 1984, P. 266.

  146. Synthesis Of 20-Dihydro-20-Deoxy Derivatives Of 16-Membered Macrolide Antibiotics ; Journal Of The Chemical Society-Chemical Communications (20): 1166-1167 1983

  147. Synthesis Of Optically-Active Penems; Journal Of The Chemical Society-Chemical Communications; (16): 908-908 1983

  148. Synthesis Of Optically-Active Penems .2. ; Tetrahedron Letters 24 (31): 3179-3182 1983

  149. Chemistry Of Natural Products, The Proceedings Of Sino-American Symposium On Chemistry Of Natural Products, Science Press, Beijing, China, P. 38 1982.

  150. New Synthesis Of Penems, The Oxalimide Cyclization Reaction ; Journal Of The American Chemical Society 104 (22): 6138-6139 1982

  151. A Stereochemical Model Of The Veratrum Alkaloids ; Journal Of Organic Chemistry 47 (21): 4137-4145 1982

  152. Chemical Degradation Of Ar-5 Antibiotics (Mycinamicins) - X-Ray Crystal-Structure Analysis Of The Aglycone From Ar-5=2 ; Journal Of The Chemical Society-Chemical Communications; (15): 853-855 1982

  153. Mutasynthesis Of 23-O-Mycinosyl-12,13-Desepoxy-12,13-Didehydrorosaramicin From Tylosin ;  Journal Of The Chemical Society-Chemical Communications ;  (15): 855-857 1982

  154. Chemical Modification Of Everninomicins ; Journal Of Antibiotics 35 (5): 561-570 1982

  155. Synthesis Of Sch-29482 - A Novel Penem Antibiotic ; Journal Of Antimicrobial Chemotherapy 9: 1-5 Suppl. C 1982

  156. A General Stereocontrolled Route To Carbocyclic C-Nucleosides - (+/-)-Carba-Showdowmycin ; Tetrahedron Letters 22 (52): 5227-5230 1981

  157. Intramolecular Cyclo-Additions Of Nitrones Joined By Amides To Olefins ; Tetrahedron 37 (21): 3615-3625 1981

  158. Synthesis Of Optically-Active Penems ; Tetrahedron Letters 22 (36): 3485-3488 1981

  159. Synthesis Of Racemic, 2-(Alkylthio)-6-(1-Hydroxyethyl) Penems - Attempted Penem Synthesis Via Copper(I) Promoted Cyclizations ; Tetrahedron Letters 22 (36): 3489-3492 1981

  160. Sch-18640 - A New Thiostrepton-Type Antibiotic ; Journal Of The American Chemical Society 103 (17): 5231-5233 1981

  161. C-13 Nmr Spectral Correlation For Simplified Structure Determination Of Curamycins And Related Oligosaccharide Antibiotics ; Heterocycles 15 (2): 1621-1641 1981

  162. Structural Elucidation Of Curamycins By Negative Chemical Ionization Mass Spectrometry, A.C.S. Meeting, San Francisco, 1980.

  163. Structure Determination Of Curamycins By Negative Chemical Ionization Mass-Spectrometry ; Abstracts Of Papers Of The American Chemical Society 180 (Aug): 374-Orgn 1980

  164. Use Of  13 C NMR To Determine Conformational Changes In Complex Antibiotic Structures, Chem. Comm., 1980.

  165. Chemical Degradation And X-Ray Crystal-Structure of Rosaramicin ; Tetrahedron Letters 21 (49): 4699-4702 1980

  166. Electrochemical Modification Of Everninomicin-D ; Journal of The Chemical Society-Chemical Communications (2): 56-58 1980

  167. X-Ray Crystal And Molecular Structure of Olgose, A Major Degradation Product Of The Oligosaccharide Antibiotic Everninomicin D, Chem. Comm., 22 1979.

  168. Current Chemotherapy And Infectious Diseases, Proc. Of The 11th Icq And The 19th Isaac, Vol. 1, 58 1979.

  169. Structural Studies On Curamycins ; Journal Of Antibiotics 32 (11): 1213-1216 1979

  170. Convenient Mass-Spectral Technique For Structural Studies On Oligosaccharides  ; Journal Of The Chemical Society-Chemical Communications (4): 148-149 1979

  171. Ansamycins, Isolation, Separation And Purification Of Antibiotics, Elsevier, 39-68 1978.

  172. Oligosaccharide Antibiotics, Encyclopedia Of Chemical Technology, 986-990 1978.

  173. Topics In Antibiotic Chemistry, Vol. 2, Oligosaccharide Antibiotics, P. 67-97, 1978.

  174. Structures Of Halomicins-A And Halomicins-C ; Journal Of Antibiotics 30 (7): 625-627 1977

  175. Stereochemistry At C-3 Of Evernitrose - Fallacy In Determination Of Stereochemistry At Quaternary Centers Using Nuclear Magnetic-Resonance Spectroscopy - X-Ray Crystal-Structure Ofmethyl 3-Acetamido-2,3,6-Trideoxy-3-C,4-O-Dimethyl-L-Xylo-Hexopyranoside ; Journal Of The Chemical Society-Chemical Communications (9): 313-314 1977

  176. Biosynthesis Of Rosamicin ; Journal Of Antibiotics 29 (9): 976-977 1976

  177. Structure Of Everninomicin-2 ; Journal Of The Chemical Society-Chemical Communications (15): 609-611 1976

  178. Electrochemical Oxidation Of Halomicin-B To Rifamycin-S ; Journal Of Organic Chemistry 41 (7): 1258-1260 1976

  179. Electrophilic Addition Of Perfluorofluoro-Oxy-Compounds To Unactivated Double-Bonds ; Journal Of The Chemical Society-Perkin Transactions 1 (1): 101-104 1976

  180. Structure Of Everninomicin-B ; Journal Of Antibiotics 28 (9): 707-709 1975

  181. Structure Of Everninomicin-C ; Journal Of Antibiotics 28 (9): 710-712 1975

  182. Structure Of Everninomicin D ; Journal Of The American Chemical Society 97 (7): 1982-1985 1975

  183. Electrophilic Fluorination Of Aromatic Substrates By Fluoroxytrifluoromethane ; Anales De Quimica 70 (12): 871-875 1974

  184. Structure Of Halomicin-B  ; Journal Of The Chemical Society-Chemical Communications (10): 395-396 1974

  185. Hydrolysis Products Of Everninomicin B ; Journal Of The Chemical Society-Chemical Communications (15): 531-532 1973

  186. Structure And Absolute Stereochemistry Of Everheptose ; Journal Of The American Chemical Society 95 (3): 942-945 1973

  187. Method For Determination Of Molecular Weights ; Journal Of The Chemical Society D-Chemical Communications (15): 823& 1971

  188. Structure Of Evertetrose And Everninonitrose ; Journal Of The Chemical Society D-Chemical Communications (14): 746& 1971

  189. Genistein And Daidzein, Metabolites Of Micromonospora-Halophytica ; Chemistry & Industry (6): 201& 1970

  190. Structure Of Evertriose, A Trisaccharide Component Of Everninomicin-D ; Journal Of The Chemical Society D-Chemical Communications (15): 911& 1970

  191. Ishwarone ; Tetrahedron 26 (10): 2371& 1970

  192. Ishwarone A Novel Tetracyclic Sesquiterpene ; Tetrahedron Letters (3): 133& 1969

  193. Structure And Absolute Stereochemistry Of Everninose, A Non-Reducing Sugar Obtained On Hydrolysis Of Everninomicin D1 ; Journal Of The Chemical Society D-Chemical Communications; (24): 1488& 1969

  194. Structure And Absolute Stereochemistry Of Evermicose ; Journal Of The Chemical Society D-Chemical Communications (19): 1149& 1969

  195. Isolation And Structure Of Surangin A And Surangin B 2 New Coumarins From Mammea Longifolia (Wight) Planch And Triana ; Tetrahedron 25 (7): 1453& 1969

  196. Organic Reactions Of Fluoroxy-Compounds – Addition Reactions Of Unactivated And Deactivated Unsaturated Linkages Of Steroids ; Journal Of The Chemical Society D-Chemical Communications (5): 227& 1969

  197. Evernitrose A Naturally Occurring Nitro Sugar From Everninomicins ; Journal Of The American Chemical Society 90 (25): 7129& 1968

  198. Organic Reactions Of Fluoroxy-Compounds – Electrophilic Fluorination Of Aromatic Rings ; Chemical Communications (14): 806& 1968

  199. Synthesis Of N-(Beta-Arylethyl)-2-Aza-3-Oxo-6-Hydroxy-Bicycl[2.2.2]Octanes ; Indian Journal Of Chemistry 6 (4): 186& 1968

  200. Chemical Investigation Of Some Indian Plants .3. ; Indian Journal Of Chemistry 5 (10): 523& 1967

  201. Synthesis Of Clausenin Xanthoxyletin Alloxanthoxyletin Xanthyletin And Nordalbergin ; Tetrahedron 23 (12): 4777& 1967

  202. Boron Trifluoride Catalysed Rearrangement Of 1,2-Epoxy Lupan-3-1; Tetrahedron 23 (9): 3847& 1967

  203. Chemical Investigation Of Some Indian Plants .2. ; Indian Journal Of Chemistry 4 (10): 457& 1966

  204. Alkaloids Of Vepris Bilocularis ; Indian Journal Of Chemistry 4 (7): 334& 1966

  205. Chemical Investigation Of Luvunga Eleutherandra ; Indian Journal Of Chemistry 4 (6): 292& 1966

  206. Oxidation Of Ring A In Lupeol, Tetrahedron, 22, 3597 1966.

  207. Structure Of Diospyrin ; Tetrahedron Letters (29): 3373& 1966

  208. Chemical Constituents Of Glochidion Hohenackeri ; Tetrahedron 22 (4): 1513& 1966

  209. Chemical Investigation Of Some Indian Plants ; Indian Journal Of Chemistry 3 (5): 237& 1965

  210. Structure Of Opuntiol A Constituent Of Opuntia Elatior ; Tetrahedron 21 (1): 93& 1965

  211. Photochemical Transformations .11. Photochemistry Of Pentacyclic Triterpenoids With Diene Unsaturation In Ring C; Journal Of The Chemical Society (Aug): 3313& 1961

  212. Leucoanthocyanidins Of Plants-Iii, J.C.S., 6, 2787 1961.

  213. Preparation Of Leucocyanidin, Current Science, 29, 53 1960.

  214. A Study Of Leucoanthocyanidins Of Plants-Ii, Tetrahedron, 6, 21 1959

  215. A Study Of Leucoanthocyanidins Of Plants-I, Tetrahedron, 3, 225 1958.

  216. Isolation Of The More Commonly Occurring Leucoanthocyanidin Of Plants, J.S.I.R., 17b, 168 1958.

  217. Synthetic Methods In The Benzo-Pyrone Series, Proc. Indian Acad. Sci., Xlvi, 19 1957.

  218. A Convenient Method Of Preparation Of Cyanidin Chloride From (+) Catechin And (-) Epicatechin, Proc. Indian Acad. Sci., Xlvi, 25 1957.